Parameterization of Org27569: An allosteric modulator of the cannabinoid CB(1) G protein-coupled receptor (full – 2011)http://www.ncbi.nlm.nih.gov/pmc/articles/PMC3145811/
Allosteric modulator ORG27569 induces CB1 cannabinoid receptor high affinity agonist binding state, receptor internalization, and Gi protein-independent ERK1/2 kinase activation (full – 2012) http://www.ncbi.nlm.nih.gov/pubmed/22343625
A key agonist-induced conformational change in the cannabinoid receptor CB1 is blocked by the allosteric ligand Org 27569 (full – 2012)http://www.ncbi.nlm.nih.gov/pmc/articles/PMC3460482/
Distinct roles of β-arrestin 1 and β-arrestin 2 in ORG27569-induced biased signaling and internalization of the cannabinoid receptor one (CB1) (full – 2013) http://www.ncbi.nlm.nih.gov/pmc/articles/PMC3617280/
Real-time characterisation of Cannabinoid Receptor 1 (CB1 ) allosteric modulators reveals novel mechanism of action (abst – 2013)http://www.ncbi.nlm.nih.gov/pubmed/23937487
Optimization of Chemical Functionalities of Indole-2-Carboxamides to Improve Allosteric Parameters for the Cannabinoid Receptor 1 (CB1) (abst – 2014) http://www.ncbi.nlm.nih.gov/pubmed/24635495
Allosteric Modulation of a Cannabinoid G Protein-coupled Receptor BINDING SITE ELUCIDATION AND RELATIONSHIP TO G PROTEIN SIGNALING (abst – 2014) http://www.jbc.org/content/289/9/582...c-2f6edbe16774
Allosteric modulator ORG27569 induces CB1 cannabinoid receptor high affinity agonist binding state, receptor internalization, and Gi protein-independent ERK1/2 kinase activation (full – 2012) http://www.ncbi.nlm.nih.gov/pubmed/22343625
A key agonist-induced conformational change in the cannabinoid receptor CB1 is blocked by the allosteric ligand Org 27569 (full – 2012)http://www.ncbi.nlm.nih.gov/pmc/articles/PMC3460482/
Distinct roles of β-arrestin 1 and β-arrestin 2 in ORG27569-induced biased signaling and internalization of the cannabinoid receptor one (CB1) (full – 2013) http://www.ncbi.nlm.nih.gov/pmc/articles/PMC3617280/
Real-time characterisation of Cannabinoid Receptor 1 (CB1 ) allosteric modulators reveals novel mechanism of action (abst – 2013)http://www.ncbi.nlm.nih.gov/pubmed/23937487
Optimization of Chemical Functionalities of Indole-2-Carboxamides to Improve Allosteric Parameters for the Cannabinoid Receptor 1 (CB1) (abst – 2014) http://www.ncbi.nlm.nih.gov/pubmed/24635495
Allosteric Modulation of a Cannabinoid G Protein-coupled Receptor BINDING SITE ELUCIDATION AND RELATIONSHIP TO G PROTEIN SIGNALING (abst – 2014) http://www.jbc.org/content/289/9/582...c-2f6edbe16774